CHEMICAL BIOLOGY & DRUG DESIGN, cilt.82, sa.4, ss.361-366, 2013 (SCI-Expanded)
Amino acid and peptide conjugates of quinine were synthesized using microwave irradiation in 52-95% yields using benzotriazole methodology. The majority of these conjugates retain in vitro antimalarial activity with IC50 values below 100nm, similar to quinine.